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Hypoglycemic Agent Screen, Serum

Test ID: HGCAS

Test

Aliases/Synonyms

Amaryl; Chlorpropamide; Dymelor; Glimepiride; Glipizide; Glucotrol; Glyburide; Meglitinides; Micronase; Prandin; Repaglinide; Sulfonylurea Hypoglycemic Serum; Sulfonylureas; Tolazamide; Tolinase; Acetohexamide ; Dymelor; Orinase ; Tolbutamide; Diabinese ; Chlorpropamide; HYPOG; Diabinese; Actoplus Met; Actos; Avandamet; Glibenclamide; Glubrava; Glucophage; Lobeglitazone; Meglitinide; Nateglinide; Novonorm; Orinase; Pioglitazone; Piomet; Politor; PPAR; Rosiglitazone; Starlix; Surepost; Thiazolidinedione; Tolazamide; Tolbutamide; Tolinase; Troglitazone; Hypoglycemic Agents

Method

Liquid Chromatography/Tandem Mass Spectrometry (LC/MS/MS)

Report Includes

Chlorpropamide; Glimepiride; Glipizide; Glyburide; Nateglinide; Pioglitazone; Repaglinide; Rosiglitazone; Tolazamide; Tolbutamide

Specimens

Serum

Clinical Utility

Evaluation of suspected insulinoma characterized by hypoglycemia and increased serum insulin concentration.
Detecting drugs that stimulate insulin secretion.
Drugs detected by this procedure are:

  • The first-generation sulfonylureas: chlorpropamide (Diabinese), tolazamide, and tolbutamide (Orinase)
  • The second-generation sulfonylureas: glimepiride (Amaryl), glipizide (Glucotrol), and glyburide (Glibenclamide)
  • The meglitinides: repaglinide (Prandin) and nateglinide (Starlix)
  • The thiazolidinediones: pioglitazone (Actos) and rosiglitazone (Avandia)

This test is not intended for therapeutic drug monitoring but could be used to monitor compliance.

Test Version

17-Nov-2025

Specimen

Specimens

Serum

Collection Containers

Red top (no additive)

Sample Volume

1.5 mL

Minimum Volume

0.5 mL

Patient Preparation

Specimen must be collected during an episode of hypoglycemia.

Stability

Ambient 7 days
Refrigerated 28 days
Frozen 28 days

Rejection Criteria

Specimen Gel-separator tubes

Test Version

17-Nov-2025

Performance / Interpretation

Method

Liquid Chromatography/Tandem Mass Spectrometry (LC/MS/MS)

Turnaround Time

8 days

Results

Name Units Reference Range Conversion Factor
Chlorpropamide
  • Negative
Screening cutoff concentration: 100 ng/mL
Glimepiride
  • Negative
Screening cutoff concentration: 20 ng/mL
Glipizide
  • Negative
Screening cutoff concentration: 5 ng/mL
Glyburide
  • Negative
Screening cutoff concentration: 5 ng/mL
Nateglinide
  • Negative
Screening cutoff concentration: 5 ng/mL
Pioglitazone
  • Negative
Screening cutoff concentration: 20 ng/mL
Repaglinide
  • Negative
Screening cutoff concentration: 5 ng/mL
Rosiglitazone
  • Negative
Screening cutoff concentration: 20 ng/mL
Tolazamide
  • Negative
Screening cutoff concentration: 50 ng/mL
Tolbutamide
  • Negative
Screening cutoff concentration: 20 ng/mL

Test Version

17-Nov-2025

Interface / Setup

HL7 Interface Codes

Order Code Result Codes Units
HGCAS 62021Tolbutamide ng/mL
62020Tolazamide ng/mL
62025Repaglinide ng/mL
64293Pioglitazone ng/mL
64292Nateglinide ng/mL
62024Glyburide ng/mL
62023Glipizide ng/mL
62022Glimepiride ng/mL
62019Chlorpropamide ng/mL
62018Acetohexamide ng/mL
64294Rosiglitazone ng/mL

Test Version

17-Nov-2025